HDM Inhibitor, 2,4-PDCA


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Cat.No.:  BSM-0145
Product Name:  HDM Inhibitor, 2,4-PDCA
CAS No.:  207671-42-9
Figure: 
Synonyms:  2,4-Pyridinecarboxylic acid, monohydrate
Description:  A histone-lysine demethylase (HKDM) inhibitor. Inhibits JARID1 proteins with an IC₅₀ values of 4.3 µM for JARID1B and 4.1 µM for JARID1A. 2, 4-PDCA does not inhibit UTX even at 10 µM.
Appearance:  White solid
Molecular Weight:  185.13
Purity:  ≥98% by titration
Storage:  -20 ̊C
Targets:  Histone lysine demethylase (HKDM)
Molecular Formula:  C₇H₅N₄ .H₂O
MDL Number:  MFCD00149413
Solubility:  DMSO
Shipping Conditions:  Gel Pack
Warning:  For Research Use Only! Not For Use in Humans.
Product Types
◆ Bioactive Small Molecules
BSM-0002 AT9283 Inquiry
◆ Cell Lines
CL-0017 Human JARID2 Knockout Cell Line 11bp deletion Inquiry
◆ Antibodies
EAb-0079 JARID2 Polyclonal Antibody Inquiry
EAb-0080 JARID1C Polyclonal Antibody Inquiry
EAb-0081 JARID1B Polyclonal Antibody Inquiry
Related Gene / Proteins
JADE1 JAK JAK1 JAK2
JAK3 JAKMIP1 JARID JARID1
JARID1A JARID1B JARID1C JARID2

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For Research Use Only. Not for use in diagnostic or therapeutic procedures.

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