| Cat.No.: | BSM-0037 |
| Product Name: | CPTH2 |
| CAS No.: | 357649-93-5 |
| Figure: |
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| Synonyms: | Cyclopentylidene-[4-(4’-chlorophenyl)thiazol-2-yl]hydrazone |
| Description: | CPTH2 is a selective inhibitor of the histone acetyltransferase Gcn5P both in vitro and in vivo (IC50 = 0.8 M). In vitro the HAT inhibitory activity of CPTH2 was caused via bridge-interaction with histone H3. In vivo it decreased acetylation of bulk histone H3 at the H3K14ac site. |
| Appearance: | White powder. |
| Molecular Weight: | 291.8 |
| Purity: | >98% (TLC); NMR (Conforms) |
| Storage: | Store desiccated as supplied at -20°C for up to 2 years. Store solutions at -20°C for up to 1 month. |
| Targets: | Gcn5P |
| Molecular Formula: | C14H14ClN3S |
| Solubility: | Dissolved in DMSO (>25 mg/ml). |
| Warning: | For Research Use Only! Not For Use in Humans. |
| Product Types | ||
| ◆ Bioactive Small Molecules | ||
| BSM-0037 | CPTH2 | Inquiry |
| BSM-0298 | CPTH2 (hydrochloride) | Inquiry |
| BSM-0299 | Butyrolactone 3 | Inquiry |
| BSM-0354 | CPTH6 (hydrobromide) | Inquiry |
| ◆ Research Kits | ||
| EKIT-0188 | GCN5 Chemiluminescent Assay Kit | Inquiry |
| Related Gene / Proteins | |||
| GCN5 | |||
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