GPCRs Class A
🧪 CXCR4-3046H
Source: HEK293
Species: Human
Tag: Non
Conjugation:
Protein Length: Met 1-Ser 352
🧪 ADRA1A-0570H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: Ser330-Val466
🧪 CCR5-0881H
Source: E.coli
Species: Human
Tag: GST
Conjugation:
Protein Length: Glu302-Leu352
🧪 CXCR4-1437H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: Ser217-Ser352
🧪 DRD2-1991H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: Lys221-Gln373
🧪 DRD5-1992H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: Asn351-His477
🧪 DRD5-1993H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: Phe361-His477
Class A GPCRs are the largest and most varied group, making up about 48% of all GPCR receptors. This class includes receptors for light, like rhodopsin, as well as key neurotransmitter receptors for dopamine and serotonin, and hormone receptors, such as adrenergic receptors. What sets Class A apart is its structure: these receptors have a short N-terminus and a specific Asp-Arg-Tyr (DRY) motif in their third transmembrane segment, which plays a crucial role in activating G-proteins. By focusing on Class A and its essential functions, we support research and innovation in areas spanning vision, mental health, and hormone-related processes.