GPCRs Class A
🧪 ADRA2A-9442H
Source: E.coli
Species: Human
Tag: GST
Conjugation:
Protein Length: 220-376a.a.

🧪 AGTRAP-9486H
Source: E.coli
Species: Human
Tag: GST
Conjugation:
Protein Length: 1-152a.a.

🧪 C5AR1-10540H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: C-term-100a.a.

🧪 CCR5-10886H
Source: E.coli
Species: Human
Tag: GST
Conjugation:
Protein Length: 257-352a.a.

🧪 CHRM1-11205H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: 210-359a.a.

🧪 DRD1-12163H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: 338-446a.a.

🧪 DRD5-12165H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: C-term-127a.a.

🧪 EDNRB-12286H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: 27-99 aa
🧪 FFAR1-12852H
Source: E.coli
Species: Human
Tag: GST
Conjugation:
Protein Length: C-term-60a.a.

🧪 FPR2-12996H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: 1-351a.a.

🧪 FSHR-13016H
Source: E.coli
Species: Human
Tag: His
Conjugation:
Protein Length: 18-352 aa
🧪 P2RY10-1495H
Source: E.coli
Species: Human
Tag:
Conjugation:
Protein Length: 171-339 aa

🧪 P2RY11-1496H
Source: E.coli
Species: Human
Tag:
Conjugation:
Protein Length: C-110aa

🧪 P2RY2-1498H
Source: E.coli
Species: Human
Tag:
Conjugation:
Protein Length: C-110aa

🧪 P2RY12-1497H
Source: E.coli
Species: Human
Tag:
Conjugation:
Protein Length: 1-342aa

Class A GPCRs are the largest and most varied group, making up about 48% of all GPCR receptors. This class includes receptors for light, like rhodopsin, as well as key neurotransmitter receptors for dopamine and serotonin, and hormone receptors, such as adrenergic receptors. What sets Class A apart is its structure: these receptors have a short N-terminus and a specific Asp-Arg-Tyr (DRY) motif in their third transmembrane segment, which plays a crucial role in activating G-proteins. By focusing on Class A and its essential functions, we support research and innovation in areas spanning vision, mental health, and hormone-related processes.